SCHEMBL23318402

SCHEMBL23318402

CN(C(=O)OC(C)(C)C)C1CCc2cc(Br)ccc2C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 10/20 0.40
KCNH2 Q12809 6/20 0.40
HTR2C P28335 4/20 0.40
NPY5R Q15761 1/20 0.39
DRD2 P14416 3/20 0.38
DRD3 P35462 2/20 0.38
DRD4 P21917 1/20 0.38
DRD1 P21728 1/20 0.38
FAAH O00519 1/20 0.36
ACHE P22303 3/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30787846 0.90 AAK1 (0.38) MCHR1NPY5R
SCHEMBL22547916 0.90 AAK1 (0.38) MCHR1NPY5R
SCHEMBL4100163 0.82 DRD3 (0.45) MCHR1DRD2DRD3DRD4
SCHEMBL4110551 0.82 DRD3 (0.45) MCHR1DRD2DRD3DRD4
SCHEMBL4100155 0.82 DRD3 (0.45) MCHR1DRD2DRD3DRD4
SCHEMBL4117256 0.81 MCHR1 (0.39) MCHR1DRD2DRD3FAAH
SCHEMBL4105102 0.81 MCHR1 (0.39) MCHR1DRD2DRD3FAAH
SCHEMBL4105094 0.81 MCHR1 (0.39) MCHR1DRD2DRD3FAAH
SCHEMBL6483133 0.80 ACHE (0.45) HTR2CACHE
SCHEMBL31730506 0.80 SRD5A1 (0.38) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021087181-A1 SUBSTITUTED PYRAZOLE COMPOUNDS AS TOLL RECEPTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-05-06 WO disclosed