SCHEMBL2332863

SCHEMBL2332863

COCC(NC(=O)OC(C)(C)C)c1nc2cc(Cl)ccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 3/20 0.49
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
LMNA P02545 3/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
GAA P10253 1/20 0.38
PYGL P06737 1/20 0.38
TRPA1 O75762 1/20 0.38
SYK P43405 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
TP53 P04637 1/20 0.37
BCHE P06276 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1479007 1.00 AAK1 (0.49) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL2326825 0.92 AAK1 (0.48) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL1479853 0.92 AAK1 (0.48) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL8481259 0.92 AAK1 (0.56) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL1481829 0.89 AAK1 (0.51) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL2332614 0.89 AAK1 (0.51) AAK1OPRM1OPRD1CTDSP1LMNA
SCHEMBL2329782 0.88 AAK1 (0.49) AAK1BCHECYP3A4CYP2C9CYP2C19
SCHEMBL1479062 0.88 AAK1 (0.49) AAK1BCHECYP3A4CYP2C9CYP2C19
SCHEMBL4157800 0.85 ALDH1A1 (0.56) AAK1LMNAALDH1A1SMN1; SMN2GAA
SCHEMBL5103994 0.84 AAK1 (0.55) AAK1OPRM1OPRD1CTDSP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771441-B1 NOVEL CARBOXAMIDES FOR USE AS XA INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2011-08-17 EP disclosed