SCHEMBL2334339

SCHEMBL2334339

COC(=O)/C=C/c1cc(F)cc(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.50
TTR P02766 1/20 0.47
APP P05067 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
TYR P14679 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
PTPN1 P18031 1/20 0.45
EPHX2 P34913 1/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
JAK2 O60674 1/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
BACE1 P56817 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2334343 1.00 AKR1C3 (0.50) AKR1C3TTRAPPCA12CA1
SCHEMBL3584119 0.88 CA12 (0.55) TTRAPPCA12CA1CA2
SCHEMBL3584118 0.88 CA12 (0.55) TTRAPPCA12CA1CA2
SCHEMBL6821064 0.88 AKR1C3 (0.56) AKR1C3TTRAPPCA12CA1
SCHEMBL6821063 0.88 AKR1C3 (0.56) AKR1C3TTRAPPCA12CA1
SCHEMBL28928255 0.83 CA12 (0.59) AKR1C3TTRAPPCA12CA1
SCHEMBL29219854 0.83 CYP3A4 (0.52) AKR1C3TTRCA12CA1CA2
SCHEMBL30671407 0.83 CYP3A4 (0.52) AKR1C3TTRCA12CA1CA2
SCHEMBL18844019 0.83 TTR (0.46) AKR1C3TTRAPPCA12CA1
SCHEMBL17705228 0.82 AKR1C3 (0.57) AKR1C3TTRAPPCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021129817-A1 PYRIMIDINE-BASED COMPOUND HAVING INHIBITORY EFFECT OF KETOHEXOKINASE (KHK) 南京明德新药研发有限公司 2021-07-01 WO disclosed
WO-2011098417-A1 SUBSTITUTED CYANOBUTYRATES HAVING HERBICIDAL ACTION BASF SE (DE) 2011-08-18 WO disclosed
US-5489592-A ALDOSE REDUCTASE INHIBITORS FOR TREATMENT OF DIABETES-RELATED DISORDERS LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1996-02-06 US disclosed