SCHEMBL2334417

SCHEMBL2334417

COc1cccc(NC(=O)C2c3cc(OC)c(OC)cc3C(=O)N(C)C2c2ccccc2F)c1.COc1cccc(NC(=O)C2c3ccccc3C(=O)N(C)C2c2cccs2)c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.59
CYP3A4 P08684 6/20 0.57
KDM4E B2RXH2 6/20 0.56
KMT2A Q03164 5/20 0.56
MEN1 O00255 3/20 0.56
NPSR1 Q6W5P4 1/20 0.56
ALDH1A1 P00352 5/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPT P10636 2/20 0.52
GLA P06280 1/20 0.52
PKM P14618 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
NPC1 O15118 1/20 0.50
CYP2C9 P11712 2/20 0.48
CYP1A2 P05177 2/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2334861 0.91 CYP3A4 (0.68) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2340254 0.90 CYP3A4 (0.69) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2338961 0.89 GAA (0.73) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2330482 0.87 GAA (0.77) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2339357 0.81 CYP3A4 (0.57) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2337039 0.79 GAA (0.60) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2337755 0.79 GAA (0.60) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2379561 0.79 GAA (0.60) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2379425 0.79 GAA (0.60) GAACYP3A4KDM4EKMT2AMEN1
SCHEMBL2336299 0.79 GAA (0.60) GAACYP3A4KDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP disclosed