SCHEMBL2340254

SCHEMBL2340254

COc1cccc(NC(=O)C2c3cc(OC)c(OC)cc3C(=O)N(C)C2c2ccccc2F)c1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.69
GAA P10253 3/20 0.64
SMN1; SMN2 Q16637 2/20 0.63
ALDH1A1 P00352 2/20 0.63
KDM4E B2RXH2 3/20 0.61
TSHR P16473 3/20 0.61
PKM P14618 1/20 0.61
KMT2A Q03164 5/20 0.56
CYP2C9 P11712 4/20 0.55
MEN1 O00255 3/20 0.55
NPC1 O15118 2/20 0.53
ALOX15 P16050 2/20 0.51
CYP1A2 P05177 3/20 0.49
MAPK1 P28482 1/20 0.49
CYP2C19 P33261 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.47
USP2 O75604 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2330482 0.91 GAA (0.77) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2334417 0.90 GAA (0.59) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2335153 0.86 GAA (0.79) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2332683 0.85 CYP3A4 (0.76) CYP3A4GAASMN1; SMN2ALDH1A1TSHR
SCHEMBL2334861 0.83 CYP3A4 (0.68) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2337751 0.83 GAA (0.74) CYP3A4GAASMN1; SMN2ALDH1A1TSHR
SCHEMBL2334030 0.81 GAA (0.82) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL2330237 0.79 GAA (0.62) CYP3A4GAAALDH1A1KDM4ETSHR
SCHEMBL2336448 0.78 GAA (1.00) CYP3A4GAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL14424953 0.76 GAA (0.71) CYP3A4GAAALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2011-09-15 US claimed
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2011-09-15 US disclosed
EP-2358682-A2 ISOQUINOLONE DERIVATIVES AS INHIBITORS OF PLAVIVIRUS REPLICATION Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2011-08-24 EP disclosed
WO-2010055164-A2 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2010-05-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224208-A1 NOVEL INHIBITORS OF FLAVIVIRUS REPLICATION MAVS, IRF3, EIF2AK2 CYP3A4 722/4885GAA 2348/4885SMN1; SMN2 4405/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.