SCHEMBL2334668

SCHEMBL2334668

Nc1nc(C(=O)N2Cc3ccccc3C2)c2cc(-c3ccccc3S(=O)(=O)N3CCCC3OC(=O)NCCO)ccc2n1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.54
HSP90AB1 P08238 3/20 0.44
ALOX5AP P20292 7/20 0.39
FEN1 P39748 7/20 0.39
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17387527 0.89 HSP90AA1 (0.56) HSP90AA1HSP90AB1ALOX5APFEN1OPRM1
SCHEMBL2509995 0.89 HSP90AA1 (0.57) HSP90AA1HSP90AB1ALOX5APFEN1
SCHEMBL17387515 0.88 HSP90AA1 (0.53) HSP90AA1HSP90AB1ALOX5APFEN1OPRM1
SCHEMBL2331903 0.86 HSP90AA1 (0.51) HSP90AA1HSP90AB1ALOX5APFEN1OPRM1
SCHEMBL901807 0.85 HSP90AA1 (0.61) HSP90AA1HSP90AB1
SCHEMBL2510626 0.83 HSP90AA1 (0.59) HSP90AA1HSP90AB1ALOX5APFEN1
SCHEMBL2512188 0.83 HSP90AA1 (0.55) HSP90AA1HSP90AB1ALOX5APFEN1
SCHEMBL17387506 0.83 HSP90AA1 (0.59) HSP90AA1HSP90AB1ALOX5APFEN1
SCHEMBL2331279 0.83 HSP90AA1 (0.59) HSP90AA1HSP90AB1ALOX5APFEN1
SCHEMBL17387508 0.83 HSP90AA1 (0.59) HSP90AA1HSP90AB1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2356110-B1 QUINAZOLINAMIDE DERIVATIVES MERCK PATENT GMBH (DE) 2016-01-06 EP claimed
EP-2356110-B1 QUINAZOLINAMIDE DERIVATIVES MERCK PATENT GMBH (DE) 2016-01-06 EP disclosed
EP-2356110-A1 QUINAZOLINAMIDE DERIVATIVES Merck Patent GmbH (DE) 2011-08-17 EP disclosed
WO-2010066324-A1 QUINAZOLINAMIDE DERIVATIVES MERCK PATENT GMBH (DE) 2010-06-17 WO disclosed