SCHEMBL23355402

SCHEMBL23355402

O=C(ONc1ccc(Oc2cccc(-c3nnc(C4CC4)o3)c2)cc1F)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
HDAC3 O15379 1/20 0.40
CYP2C9 P11712 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MAPT P10636 2/20 0.39
TNKS O95271 6/20 0.37
PARP2 Q9UGN5 5/20 0.37
PARP1 P09874 4/20 0.37
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
ALDH1A1 P00352 1/20 0.36
DHODH Q02127 1/20 0.36
BRAF P15056 2/20 0.36
KDR P35968 2/20 0.36
LCLAT1 Q6UWP7 1/20 0.35
TP53 P04637 1/20 0.35
NR1H4 Q96RI1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23355377 0.86 KDM4E (0.44) KDM4EMAPTTNKSPARP2PARP1
SCHEMBL23355454 0.83 SMN1; SMN2 (0.39) KDM4EMAPTALDH1A1DHODHLCLAT1
SCHEMBL23368199 0.81 KDM4E (0.40) KDM4EMAPTTNKSPARP2PARP1
SCHEMBL30203050 0.81 KDM4E (0.40) KDM4EMAPTTNKSPARP2PARP1
Trifluoroacetic Acid SCHEMBL23355399 0.81 KDM4E (0.45) KDM4EHDAC3CYP2C9HDAC1HDAC6
SCHEMBL23368034 0.77 KDM4E (0.50) KDM4EMAPTBACE1BACE2ALDH1A1
SCHEMBL23355465 0.75 GSK3B (0.37) KDM4EHDAC3HDAC1HDAC6DHODH
SCHEMBL23355403 0.74 KDM4E (0.40) KDM4EHDAC1HDAC6ALDH1A1DHODH
SCHEMBL21612784 0.72 KDM4E (0.47) KDM4EMAPTTNKSPARP2PARP1
SCHEMBL23355373 0.71 KDM4E (0.45) KDM4EMAPTALDH1A1DHODHLCLAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed