SCHEMBL23355403

SCHEMBL23355403

Cc1nnc(-c2cccc(Oc3ccc(NOC(=O)C(F)(F)F)c(F)c3)c2)s1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
HSD17B10 Q99714 4/20 0.40
HPGD P15428 4/20 0.40
ALDH1A1 P00352 2/20 0.40
USP2 O75604 1/20 0.40
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
HDAC6 Q9UBN7 4/20 0.35
FGFR3 P22607 1/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 3/20 0.35
DHODH Q02127 1/20 0.35
GAA P10253 1/20 0.35
ESR1 P03372 1/20 0.34
POLB P06746 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC1 Q13547 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23355412 0.86 KDM4E (0.47) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
SCHEMBL23368104 0.81 KDM4E (0.45) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
SCHEMBL30203359 0.81 KDM4E (0.45) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
Trifluoroacetic Acid SCHEMBL23355400 0.79 KDM4E (0.40) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
SCHEMBL23355465 0.78 GSK3B (0.37) KDM4ESMN1; SMN2HDAC6DHODHHDAC1
SCHEMBL23355454 0.77 SMN1; SMN2 (0.39) KDM4ESMN1; SMN2HPGDALDH1A1KMT2A
SCHEMBL23368055 0.74 SMN1; SMN2 (0.45) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
SCHEMBL23355402 0.74 KDM4E (0.41) KDM4EALDH1A1HDAC6DHODHHDAC1
SCHEMBL21612819 0.70 NOTUM (0.40) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1
SCHEMBL23355373 0.65 KDM4E (0.45) KDM4ESMN1; SMN2HSD17B10HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed