SCHEMBL23355446

SCHEMBL23355446

NC(=O)Oc1ccc(Oc2nc(CO)cs2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.36
PRSS1 P07477 1/20 0.34
TMPRSS15 P98073 1/20 0.34
FFAR1 O14842 3/20 0.31
PPARD Q03181 3/20 0.31
ICAM1 P05362 1/20 0.31
SELE P16581 1/20 0.31
SLC8A1 P32418 1/20 0.31
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
GCK P35557 1/20 0.31
SCN4A P35499 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21612851 0.87 SCN9A (0.35) SCN9APRSS1TMPRSS15
SCHEMBL23355321 0.77 GCK (0.32) PRSS1TMPRSS15ICAM1SELEGCK
SCHEMBL28527025 0.76
SCHEMBL28523464 0.75 MEN1 (0.38) FFAR1PPARDALDH1A1SCN4A
SCHEMBL23355323 0.75 MEN1 (0.40) PPARDALDH1A1
SCHEMBL23355478 0.72 MAPT (0.34) SCN9A
SCHEMBL23355451 0.72 CYP17A1 (0.42) SCN9A
SCHEMBL23368138 0.71 HSD17B10 (0.47) SCN9AGAAKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL30203152 0.71 HSD17B10 (0.46) SCN9AGAAKDM4EALDH1A1HPGD
SCHEMBL16399169 0.69 NPC1 (0.44) SCN9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed
CN-112334460-A Biaryl ether type quinazoline derivative 第一三共株式会社 2021-02-05 CN disclosed