SCHEMBL23368030

SCHEMBL23368030

CC(C)(C)OC(=O)Nc1ccc(Oc2cccc(Br)c2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
LMNA P02545 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
NPSR1 Q6W5P4 3/20 0.45
CYP3A4 P08684 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2D6 P10635 1/20 0.45
ATM Q13315 1/20 0.45
CYP17A1 P05093 1/20 0.44
AAK1 Q2M2I8 3/20 0.43
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KMT2A Q03164 1/20 0.40
P2RY1 P47900 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30203084 1.00 NPC1 (0.46) NPC1RAB9ASMN1; SMN2LMNANFKB1
SCHEMBL23368165 0.88 RAB9A (0.47) NPC1RAB9ASMN1; SMN2LMNANPSR1
SCHEMBL21612816 0.85 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNANPSR1
SCHEMBL23355361 0.85 NPC1 (0.49) NPC1RAB9ASMN1; SMN2CYP2C9CYP17A1
SCHEMBL23355337 0.84 SMN1; SMN2 (0.47) NPC1RAB9ASMN1; SMN2LMNANFKB1
SCHEMBL64834 0.83 AAK1 (0.53) NPC1RAB9ASMN1; SMN2LMNANFKB1
SCHEMBL30203283 0.83 KCNQ4 (0.43) NPC1RAB9ASMN1; SMN2NPSR1CYP17A1
SCHEMBL23368045 0.83 KCNQ4 (0.43) NPC1RAB9ASMN1; SMN2NPSR1CYP17A1
SCHEMBL23355301 0.82 NPC1 (0.48) NPC1RAB9ASMN1; SMN2LMNANFKB1
SCHEMBL23368134 0.82 RAB9A (0.48) NPC1RAB9ASMN1; SMN2LMNANFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822263-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2021-05-19 EP disclosed