SCHEMBL23385355

SCHEMBL23385355

C=C(Nc1cnc(Cl)cc1-c1ccc(F)cc1C)C(C)(C)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.53
TACR1 P25103 15/20 0.41
CYP3A4 P08684 9/20 0.41
TACR3 P29371 7/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30980992 0.88 GPBAR1 (0.58) GPBAR1TACR1CYP3A4TACR3
SCHEMBL23361960 0.88 GPBAR1 (0.58) GPBAR1TACR1CYP3A4TACR3
SCHEMBL337412 0.78 GPBAR1 (0.54) GPBAR1TACR1CYP3A4TACR3
SCHEMBL336672 0.75 GPBAR1 (0.51) GPBAR1TACR1CYP3A4TACR3
SCHEMBL336998 0.75 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL30981004 0.75 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL30981003 0.75 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL1872308 0.73 GPBAR1 (0.46) GPBAR1
SCHEMBL1872544 0.73 GPBAR1 (0.74) GPBAR1TACR1CYP3A4TACR3
SCHEMBL336870 0.73 GPBAR1 (0.48) GPBAR1TACR1CYP3A4TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021094247-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2021-05-20 WO disclosed