SCHEMBL30980992

SCHEMBL30980992

Cc1cc(F)ccc1-c1cc(Cl)ncc1NC(=O)C(C)(C)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.58
TACR1 P25103 15/20 0.46
CYP3A4 P08684 9/20 0.44
TACR3 P29371 6/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23361960 1.00 GPBAR1 (0.58) GPBAR1TACR1CYP3A4TACR3
SCHEMBL23385355 0.88 GPBAR1 (0.53) GPBAR1TACR1CYP3A4TACR3
SCHEMBL337412 0.82 GPBAR1 (0.54) GPBAR1TACR1CYP3A4TACR3
SCHEMBL336998 0.79 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL30981003 0.79 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL30981004 0.79 GPBAR1 (0.77) GPBAR1TACR1CYP3A4TACR3
SCHEMBL336672 0.79 GPBAR1 (0.51) GPBAR1TACR1CYP3A4TACR3
SCHEMBL16708969 0.78 TACR1 (0.48) GPBAR1TACR1CYP3A4TACR3
SCHEMBL1872544 0.77 GPBAR1 (0.74) GPBAR1TACR1CYP3A4TACR3
SCHEMBL16001625 0.77 TACR1 (0.46) TACR1CYP3A4TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114728906-B Novel chemical process for preparing the key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridin-3-amine of NT-814 康堤医疗有限公司 2024-08-20 CN claimed
CN-118496152-A Novel chemical process for preparing the key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridin-3-amine of NT-814 康堤医疗有限公司 2024-08-16 CN claimed
CN-114728906-B Novel chemical process for preparing the key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridin-3-amine of NT-814 康堤医疗有限公司 2024-08-20 CN disclosed
CN-118496152-A Novel chemical process for preparing the key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridin-3-amine of NT-814 康堤医疗有限公司 2024-08-16 CN disclosed