SCHEMBL23394

SCHEMBL23394

CNc1nc2c(Cl)nccn2n1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.32
HTR6 P50406 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24659 0.83
SCHEMBL15221252 0.81 PDE10A (0.38) FLT3HTR6
SCHEMBL19266 0.77 KDR (0.48)
SCHEMBL20035 0.76 JAK2 (0.51)
SCHEMBL15210382 0.74 JAK2 (0.53)
SCHEMBL20918 0.74 FLT1 (0.42)
SCHEMBL16394606 0.74 CDK19 (0.44) FLT3
SCHEMBL15221144 0.74 JAK2 (0.46)
SCHEMBL21018 0.73 NFKB1 (0.51)
SCHEMBL15221233 0.73 JAK2 (0.60) FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817310-B1 8-SUBSTITUTED 2-AMINO-[1,2,4]TRIAZOLO[1,5-A]PYRAZINES AS SYK TRYROSINE KINASE INHIBITORS AND GCN2 SERIN KINASE INHIBITORS MERCK PATENT GMBH (DE) 2018-03-21 EP disclosed
WO-2012025186-A1 TRIAZOLOPYRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-03-01 WO disclosed