SCHEMBL2340306

SCHEMBL2340306

CC(C)(CO)CNC(=O)Oc1c[nH]c2ncc(-c3cccs3)nc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.36
NOS1 P29475 1/20 0.35
SYK P43405 3/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 2/20 0.34
ADORA2A P29274 4/20 0.34
ADORA3 P0DMS8 3/20 0.34
ADORA1 P30542 3/20 0.34
MAPT P10636 3/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
MAPK10 P53779 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1370911 0.84 SYK (0.45) SYKCYP2D6TSHR
SCHEMBL2351523 0.78 SYK (0.54) SYK
SCHEMBL2344786 0.78 JAK2 (0.48)
SCHEMBL18524459 0.75 SYK (0.61) SYK
SCHEMBL2344505 0.74 MAP4K1 (0.36) ATRSYKCYP2D6TSHRMEN1
SCHEMBL1896593 0.73 JAK3 (0.49) NOS1SYKCYP2D6MAPTMEN1
SCHEMBL1889903 0.70 SYK (0.39) ATRNOS1SYKCYP2D6MAPT
SCHEMBL3395862 0.70 KDM4E (0.48) NOS1MEN1KMT2ANPC1RAB9A
SCHEMBL1368571 0.69 ERCC1 (0.47) NOS1SYKCYP2D6ADORA2AADORA3
SCHEMBL1368569 0.69 JAK3 (0.57) SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247592-B1 PYRROLOPYRAZINE KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2011-08-31 EP claimed