SCHEMBL23428958

SCHEMBL23428958

Cc1cccc(C(NC[C@H]2CCCO2)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
HPGD P15428 5/20 0.52
GAA P10253 2/20 0.50
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
PKM P14618 2/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.46
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17073448 0.80 TACR1 (0.47) RAB9ACYP3A4
SCHEMBL23429069 0.75 KLKB1 (0.44) NPC1
SCHEMBL23429132 0.74 SIGMAR1 (0.43)
SCHEMBL3397976 0.72 HPGD (0.43) ALDH1A1HPGDRAB9APKMCYP3A4
SCHEMBL9185050 0.71 MTOR (0.52) ALDH1A1HPGDRAB9APKMCYP3A4
SCHEMBL9729131 0.71 HPGD (0.55) ALDH1A1HPGDGAARAB9APKM
SCHEMBL14492278 0.71 ATM (0.70) HPGDGAANPC1RAB9APKM
SCHEMBL17073430 0.70 KLKB1 (0.42) ALDH1A1NPC1
SCHEMBL23429097 0.70 GAA (0.50) ALDH1A1HPGDGAANPC1RAB9A
SCHEMBL25665861 0.70 GAA (0.50) ALDH1A1HPGDGAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4180424-A1 SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS BioCryst Pharmaceuticals, Inc. (US) 2023-05-17 EP disclosed
EP-3828173-A1 SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS BioCryst Pharmaceuticals, Inc. (US) 2021-06-02 EP disclosed