SCHEMBL23456802

SCHEMBL23456802

COc1cc2nccc(Oc3ccc(NC(=O)c4nn(CCN)cc4OCC(F)(F)F)c(F)c3)c2cc1OC

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.56
AXL P30530 5/20 0.56
PDGFRA P16234 4/20 0.56
FGFR2 P21802 2/20 0.56
KIT P10721 1/20 0.56
MET P08581 8/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23456935 0.95 KDR (0.57) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23456797 0.94 MET (0.57) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23457007 0.94 KDR (0.56) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23457199 0.93 KDR (0.55) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23456823 0.91 KDR (0.59) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23457196 0.91 KDR (0.55) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23457011 0.90 AXL (0.53) KDRAXLPDGFRAKITMET
SCHEMBL23456975 0.90 KDR (0.55) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23457122 0.90 KDR (0.51) KDRAXLPDGFRAFGFR2KIT
SCHEMBL23458667 0.88 KDR (0.53) KDRAXLPDGFRAFGFR2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210163448-A1 QUINOLINE DERIVATIVES AS INHIBITORS OF AXL/MER RTK AND CSF1R QURIENT CO., LTD. (KR) 2021-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210163448-A1 QUINOLINE DERIVATIVES AS INHIBITORS OF AXL/MER RTK AND CSF1R CSF1R, CSF3R, FLT3 KDR 25/4885AXL 4/4885PDGFRA 41/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.