SCHEMBL2345902

SCHEMBL2345902

Cc1nnc(N(c2nc(Cc3ccc(Cl)cc3)cc(C(C)(C)O)n2)C2CCNCC2)o1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 4/20 0.49
PSEN2 P49810 4/20 0.49
APH1B Q8WW43 4/20 0.49
NCSTN Q92542 4/20 0.49
APH1A Q96BI3 4/20 0.49
PSENEN Q9NZ42 4/20 0.49
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
PLAT P00750 2/20 0.33
KCNH2 Q12809 1/20 0.31
HTR6 P50406 1/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SHMT1 P34896 1/20 0.31
SHMT2 P34897 1/20 0.31
PDE6D O43924 1/20 0.30
SSTR4 P31391 1/20 0.30
THRB P10828 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14312136 0.81 PSEN1 (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2347405 0.77 P2RY14 (0.35) HTR2CPLATSLC6A2SLC6A4
SCHEMBL2269500 0.70 PSEN1 (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2354817 0.67 IKBKB (0.32)
SCHEMBL2278329 0.67 PSEN1 (0.77) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL2273652 0.65 PSEN1 (0.49) PSEN1PSEN2APH1BNCSTNAPH1A
Tert-Butyl Formate SCHEMBL27913074 0.64 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5763935 0.61 PRCP (0.45) HTR2CHTR2BPLATKCNH2HTR6
Hydrochloric Acid SCHEMBL5765388 0.60 PRCP (0.44) HTR2CHTR2BPLATKCNH2HTR6
Hydrochloric Acid SCHEMBL12078705 0.60 PSEN1 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536710-A2 PIPERIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-12-26 EP disclosed
WO-2011101304-A2 PIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-25 WO disclosed