SCHEMBL2347405

SCHEMBL2347405

Cc1nnc(N(c2nc(-c3ccc(C(F)(F)F)cc3)cc(C(C)(C)O)n2)C2CCNCC2)o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 7/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
PAX8 Q06710 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ADORA3 P0DMS8 1/20 0.31
SCN9A Q15858 2/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
NOTUM Q6P988 1/20 0.31
ADRB3 P13945 2/20 0.31
ADRA2B P18089 2/20 0.31
DRD1 P21728 2/20 0.31
DRD5 P21918 2/20 0.31
ADRA1B P35368 2/20 0.31
TMEM97 Q5BJF2 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2351952 0.80 SYK (0.35) P2RY14MEN1GAAMAPTMAPK1
SCHEMBL14312081 0.80 P2RY14 (0.35) P2RY14MEN1GAAMAPTMAPK1
SCHEMBL2345902 0.77 PSEN1 (0.49) SLC6A2SLC6A4PLATHTR2C
SCHEMBL2354817 0.71 IKBKB (0.32) MEN1MAPTMAPK1KMT2A
SCHEMBL2276128 0.68 PSEN1 (0.46) MAPTMAPK1SCN9ASYK
SCHEMBL2271701 0.64 CASP1 (0.44) MEN1MAPTKMT2ANPSR1ADORA3
SCHEMBL3408049 0.60 PTGS2 (0.46) ADORA3SYK
SCHEMBL3412138 0.60 PTGS2 (0.45) SYK
SCHEMBL6403119 0.57 NPC1 (0.55) MEN1KMT2ANPSR1NOTUM
SCHEMBL3544007 0.57 MEN1 (0.68) MEN1MAPK1KMT2ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536710-A2 PIPERIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-12-26 EP disclosed
WO-2011101304-A2 PIPERIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-25 WO disclosed