SCHEMBL23466751

SCHEMBL23466751

COC(=O)c1ccc(NC(=O)C(N)Cc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.60
NPC1 O15118 1/20 0.60
GAA P10253 2/20 0.59
L3MBTL1 Q9Y468 2/20 0.59
ALDH1A1 P00352 2/20 0.59
LNPEP Q9UIQ6 6/20 0.57
LMNA P02545 2/20 0.56
MAPT P10636 2/20 0.56
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
BACE1 P56817 2/20 0.55
SLC7A5 Q01650 1/20 0.54
HTT P42858 1/20 0.54
ERAP2 Q6P179 2/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HDAC8 Q9BY41 1/20 0.52
ROCK2 O75116 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23466750 1.00 RAB9A (0.60) RAB9ANPC1GAAL3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL29758042 0.99 RAB9A (0.59) RAB9ANPC1GAAL3MBTL1ALDH1A1
SCHEMBL19805597 0.88 MAPT (0.60) RAB9ANPC1GAAALDH1A1MAPT
SCHEMBL28753025 0.88 MAPT (0.60) RAB9ANPC1GAAALDH1A1MAPT
SCHEMBL8120133 0.88 SLC7A5 (0.56) ALDH1A1LNPEPLMNABACE1SLC7A5
SCHEMBL2995175 0.87 SLC7A5 (0.56) RAB9ANPC1LNPEPBACE1SLC7A5
SCHEMBL2995178 0.87 SLC7A5 (0.56) RAB9ANPC1LNPEPBACE1SLC7A5
SCHEMBL23486647 0.87 NAMPT (0.55) GAAL3MBTL1ALDH1A1LNPEPMAPT
Hydrochloric Acid SCHEMBL23466585 0.86 SLC7A5 (0.55) RAB9ANPC1LNPEPBACE1SLC7A5
SCHEMBL2994483 0.86 BACE1 (0.57) RAB9ANPC1BACE1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114539158-B FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2023-12-08 CN disclosed
CN-114539158-A FXIa inhibitor compound and preparation method and application thereof 沈阳药科大学 2022-05-27 CN disclosed
CN-109721539-B Pyrazole amide derivative and preparation method and application thereof 天津药物研究院有限公司 2021-07-09 CN disclosed
WO-2021110076-A1 OXAMIDE DERIVATIVES, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 深圳信立泰药业股份有限公司 2021-06-10 WO disclosed
CN-109721539-A Pyrazole amide analog derivative and its preparation method and application 天津药物研究院有限公司 2019-05-07 CN disclosed