SCHEMBL2347737

SCHEMBL2347737

CCCCc1nnc(OC2CCN(C)CC2C)cc1-c1ccc(OC2CCCCC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.35
ACVR1 Q04771 1/20 0.35
CTSL P07711 2/20 0.34
CTSB P07858 2/20 0.34
CTSS P25774 2/20 0.34
CYP2D6 P10635 1/20 0.33
AGER Q15109 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
SCN1A P35498 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN3A Q9NY46 1/20 0.32
DDX3X O00571 1/20 0.32
APP P05067 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
GRM2 Q14416 1/20 0.31
BTK Q06187 1/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12254297 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2348986 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2383098 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2348979 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2382089 0.90 TGFBR1 (0.40) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2382115 0.90 TGFBR1 (0.40) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL2382093 0.90 TGFBR1 (0.40) TGFBR1ACVR1CTSLCTSBCTSS
SCHEMBL12254293 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
Hydrochloric Acid SCHEMBL2352956 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS
Hydrochloric Acid SCHEMBL2349370 0.90 TGFBR1 (0.35) TGFBR1ACVR1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536283-A1 PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF TransTech Pharma, Inc (US) 2012-12-26 EP disclosed
WO-2011103091-A1 PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF TRANSTECH PHARMA, INC. (US) 2011-08-25 WO disclosed