SCHEMBL2348058

SCHEMBL2348058

CC(C)C[C@H](NCc1cccc(-c2cc(C(N)=O)c(NC(N)=O)s2)c1)C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.52
JAK2 O60674 2/20 0.52
JAK3 P52333 1/20 0.52
CHEK1 O14757 9/20 0.48
MEN1 O00255 1/20 0.45
EIF2AK2 P19525 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1148139 0.90 IKBKB (0.55) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL29588779 0.90 IKBKB (0.55) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL2281680 0.88 IKBKB (0.60) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL2281654 0.88 IKBKB (0.60) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL2282387 0.85 CHEK1 (0.54) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL2282382 0.85 CHEK1 (0.54) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL11921317 0.84 IKBKB (0.59) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL10166372 0.83 ALDH1A1 (0.43) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL560462 0.83 ALDH1A1 (0.43) IKBKBJAK2JAK3CHEK1MEN1
SCHEMBL2347803 0.83 CHEK1 (0.49) IKBKBJAK2JAK3CHEK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078007-B1 IKK-BETA SERINE-THREONINE PROTEIN KINASE INHIBITORS CHROMA THERAPEUTICS LTD (GB) 2011-08-31 EP claimed