SCHEMBL23486299

SCHEMBL23486299

Cc1ccc(Cc2cccc(C#N)c2)cc1C#N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
GLA P06280 1/20 0.44
SCN8A Q9UQD0 1/20 0.43
FFAR1 O14842 2/20 0.41
TSHR P16473 1/20 0.40
CYP19A1 P11511 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
MPO P05164 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38
TP53 P04637 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
MEP1A Q16819 1/20 0.38
MEP1B Q16820 1/20 0.38
ERCC1 P07992 1/20 0.37
ERCC4 Q92889 1/20 0.37
MAOB P27338 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.37
KLKB1 P03952 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12113905 0.86 TSHR (0.46) FFAR1TSHRLOXL2
SCHEMBL2153847 0.82 HRH3 (0.59) IDH1HRH3GLAFFAR1TSHR
SCHEMBL23958863 0.79 FFAR1 (0.46) IDH1FFAR1TSHRFFAR4LOXL2
SCHEMBL4196662 0.77 HRH3 (0.54) IDH1HRH3GLAFFAR1TSHR
SCHEMBL7626603 0.75 CLK4 (0.47) TSHR
SCHEMBL26987873 0.75 HRH3 (0.49) IDH1HRH3GLAFFAR1CYP19A1
SCHEMBL481239 0.75 HRH3 (0.49) IDH1HRH3GLAFFAR1CYP19A1
SCHEMBL1003188 0.74 TSHR (0.50) FFAR1TSHRCYP11B1CYP11B2FFAR4
SCHEMBL18609498 0.74 IDH1 (0.47) IDH1HRH3GLASCN8ACYP19A1
SCHEMBL18641315 0.74 LTA4H (0.58) IDH1HRH3GLAFFAR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021113263-A1 CRF RECEPTOR ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES, INC. (US) 2021-06-10 WO disclosed