SCHEMBL23532503

SCHEMBL23532503

C=CCOC(=O)N(CC=C)CC(OC)OC

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TSHR P16473 1/20 0.33
CYP3A4 P08684 1/20 0.31
LMNA P02545 1/20 0.31
DPP4 P27487 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8741042 0.87 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ALMNADPP4
SCHEMBL1683063 0.80 ALDH1A1 (0.45) TDP1ALDH1A1MEN1KMT2ATSHR
SCHEMBL9178860 0.80 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ALMNADPP4
SCHEMBL654305 0.78 ALDH1A1 (0.42) TDP1ALDH1A1KMT2A
SCHEMBL28320454 0.78 ALDH1A1 (0.40) TDP1ALDH1A1CYP3A4LMNA
SCHEMBL17688553 0.78 ALDH1A1 (0.39) TDP1ALDH1A1MEN1KMT2ATSHR
SCHEMBL7252003 0.75 ALDH1A1 (0.41) TDP1ALDH1A1TSHRCYP3A4
SCHEMBL9874189 0.75 ALDH1A1 (0.35) ALDH1A1MEN1KMT2ALMNADPP4
SCHEMBL10537484 0.75 TSHR (0.37) TDP1ALDH1A1MEN1KMT2ATSHR
SCHEMBL23532412 0.74 ALDH1A1 (0.39) TDP1ALDH1A1TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021123785-A1 DNA POLYMERASE THETA INHIBITORS ARTIOS PHARMA LIMITED (GB) 2021-06-24 WO disclosed
WO-2021123785-A1 DNA POLYMERASE THETA INHIBITORS ARTIOS PHARMA LIMITED (GB) 2021-06-24 WO disclosed