SCHEMBL2353368

SCHEMBL2353368

COC(=O)[C@H]1CC(O[Si](C)(C)C(C)(C)C)C(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.34
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
MMP2 P08253 1/20 0.32
ANPEP P15144 1/20 0.32
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
PDE4B Q07343 1/20 0.31
P2RX3 P56373 1/20 0.31
IMPDH2 P12268 3/20 0.30
KAT2B Q92831 1/20 0.30
USP2 O75604 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31234416 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL2494729 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL18204848 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL2494727 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL12192438 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL15122945 1.00 PTPN1 (0.34) PTPN1NR1H2NR1H3MMP2ANPEP
SCHEMBL15133204 0.89 CHRM2 (0.32) NR1H2CHRM2CHRM1CHRM3USP2
SCHEMBL20380929 0.87 GLA (0.34) NR1H2
SCHEMBL18612437 0.87 GLA (0.34) NR1H2
SCHEMBL5455578 0.86 MAPT (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100010234-A1 PROCESS FOR MANUFACTURING A GLUTAMIC ACID DERIVATIVE AND A PYROGLUTAMIC ACID DERIVATIVE AND A NOVEL INTERMEDIATE IN THE MANUFACTURE THEREOF AJINOMOTO CO. INC (JP) 2010-01-14 US claimed
US-20060009394-A1 Process for manufacturing a glutamic acid derivative and a pyroglutamic acid derivative and a novel intermediate in the manufacture thereof AJINOMOTO CO. INC (JP) 2006-01-12 US claimed
US-8394970-B2 Process for manufacturing a glutamic acid derivative and a pyroglutamic acid derivative and a novel intermediate in the manufacture thereof AJINOMOTO CO., INC. (JP) 2013-03-12 US disclosed
EP-1582514-B1 PROCESSES FOR PRODUCING GLUTAMIC ACID DERIVATIVE, A PYROGLUTAMIC ACID DERIVATIVE AND A NOVEL INTERMEDIATE FOR PRODUCTION AJINOMOTO KK (JP) 2011-08-31 EP disclosed
US-7674915-B2 Process for manufacturing a glutamic acid derivative and a pyroglutamic acid derivative and a novel intermediate in the manufacture thereof AJINOMOTO CO., INC. (JP) 2010-03-09 US disclosed
US-20100010234-A1 PROCESS FOR MANUFACTURING A GLUTAMIC ACID DERIVATIVE AND A PYROGLUTAMIC ACID DERIVATIVE AND A NOVEL INTERMEDIATE IN THE MANUFACTURE THEREOF AJINOMOTO CO. INC (JP) 2010-01-14 US disclosed
US-20060009394-A1 Process for manufacturing a glutamic acid derivative and a pyroglutamic acid derivative and a novel intermediate in the manufacture thereof AJINOMOTO CO. INC (JP) 2006-01-12 US disclosed
EP-1582514-A1 PROCESSES FOR PRODUCING GLUTAMIC ACID DERIVATIVE AND PYROGLUTAMIC ACID DERIVATIVE AND NOVEL INTERMEDIATE FOR PRODUCTION Ajinomoto Co., Inc. (JP) 2005-10-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100010234-A1 PROCESS FOR MANUFACTURING A GLUTAMIC ACID DERIVATIVE AND A PYROGLUTAMIC ACID DERIVATIVE AND A NOVEL INTERMEDIATE IN THE MANUFACTURE THEREOF PTMA, GRIK5, GLUL PTPN1 4780/4885NR1H2 4627/4885NR1H3 4593/4885
US-20060009394-A1 Process for manufacturing a glutamic acid derivative and a pyroglutamic acid derivative and a novel intermediate in the manufacture thereof PTMA, GRIK5, GLUL PTPN1 4780/4885NR1H2 4627/4885NR1H3 4593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.