SCHEMBL23535

SCHEMBL23535

CC1(C)CCNC1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 5/20 0.49
DPP4 P27487 2/20 0.45
PITRM1 Q5JRX3 2/20 0.45
DPP9 Q86TI2 2/20 0.45
FAP Q12884 1/20 0.45
DPP8 Q6V1X1 1/20 0.45
DPP7 Q9UHL4 1/20 0.45
APLNR P35414 1/20 0.34
CYP2D6 P10635 2/20 0.33
LMNA P02545 2/20 0.33
BLM P54132 2/20 0.33
TSHR P16473 2/20 0.33
PMP22 Q01453 2/20 0.33
ALOX15 P16050 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
FFAR3 O14843 1/20 0.33
MEN1 O00255 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536 1.00 ARG1 (0.49) ARG1DPP4PITRM1DPP9FAP
Hydrochloric Acid SCHEMBL16393846 0.98 ARG1 (0.47) ARG1DPP4PITRM1DPP9FAP
Hydrochloric Acid SCHEMBL905291 0.98 ARG1 (0.47) ARG1DPP4PITRM1DPP9FAP
Hydrochloric Acid SCHEMBL905290 0.98 ARG1 (0.47) ARG1DPP4PITRM1DPP9FAP
SCHEMBL9187521 0.87 DPP4 (0.49) ARG1DPP4PITRM1DPP9FAP
SCHEMBL27561362 0.85 DPP4 (0.44) ARG1DPP4PITRM1DPP9FAP
Hydrochloric Acid SCHEMBL31389556 0.85 DPP4 (0.48) ARG1DPP4PITRM1DPP9FAP
SCHEMBL8894788 0.82 CYP2D6 (0.40) ARG1DPP4PITRM1DPP9FAP
SCHEMBL4209356 0.80 ARG1 (0.47) ARG1DPP4PITRM1DPP9FAP
SCHEMBL1485387 0.80 DPP4 (0.44) ARG1DPP4PITRM1DPP9FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2824 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11203622-B2 MASP isoforms as inhibitors of complement activation OMEROS CORPORATION (US) 2021-12-21 US claimed
WO-2005026114-A1 HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME AND THEIR PHARMACEUTICAL USES PFIZER INC. (US) 2005-03-24 WO claimed
US-6329502-B1 VIRICIDES AGAINST HUMAN IMMUNODEFICIENCY VIRUS; TREATMENT OF AIDS (ACQUIRED IMMUNE DEFICIENCY SYNDROME) JAPAN ENERGY CORPORATION (JP) 2001-12-11 US claimed
US-6313094-B1 COMPOSITION FOR INHIBITING HUMAN IMMUNODEFICIENCY VIRUS REPLICATION JAPAN ENERGY CORPORATION (JP) 2001-11-06 US claimed
US-6084065-A FOR AGRICULTURAL USE ISAGRO SPA (IT) 2000-07-04 US claimed
EP-0956293-A1 THROMBIN INHIBITORS Akzo Nobel N.V. (NL) 1999-11-17 EP claimed
EP-0490667-B1 HIV protease inhibitors JAPAN ENERGY CORP (JP) 1999-06-09 EP claimed
WO-1998007308-A2 THROMBIN INHIBITORS AKZO NOBEL N.V. (NL) 1998-02-26 WO claimed
US-5698672-A ADMINSTERING TO TREAT OSTEOPOROSIS, PAGET'S DISEASE AND HYPERPARATHYROIDISM ZYMOGENETICS, INC. (US) 1997-12-16 US claimed
WO-1996031536-A1 SYNTHETIC CALCITONIN MIMETICS ZYMOGENETICS, INC. (US) 1996-10-10 WO claimed
EP-0652229-A2 Oligopeptides with fungicidal activity ISAGRO S.p.A. (IT) 1995-05-10 EP claimed
EP-0422937-B1 Fibrinogen receptor antagonists MERCK & CO INC (US) 1994-03-02 EP claimed
WO-1993000108-A1 NOVEL INHIBITORS OF PLATELET AGGREGATION CORVAS INTERNATIONAL, INC. (US) 1993-01-07 WO claimed
EP-0490667-A2 HIV protease inhibitors JAPAN ENERGY CORPORATION (JP) 1992-06-17 EP claimed
US-5023233-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1991-06-11 US claimed
EP-0411833-A1 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1991-02-06 EP claimed
EP-0410539-A1 Fibrinogen receptor antagonists MERCK & CO. INC. (US) 1991-01-30 EP claimed
US-20260062449-A1 PEPTIDE COMPOSITIONS AND METHODS OF USE ONL THERAPEUTICS INC (US) 2026-03-05 US disclosed
US-4691022-A Process for the preparation of monocyclic, bicyclic and tricyclic aminoacids HOECHST AKTIENGESELLSCHAFT (DE) 1987-09-01 US disclosed
EP-0132580-A1 Process for the preparation of mono, bi and tricyclic aminoacids HOECHST AKTIENGESELLSCHAFT (DE) 1985-02-13 EP disclosed