SCHEMBL2356095

SCHEMBL2356095

Cc1ccc(-n2nccn2)c(C(=O)N2CCOCC2)c1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.58
HCRTR1 O43613 19/20 0.58
CYP3A4 P08684 7/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17501812 0.88 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL17539262 0.86 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL2358754 0.86 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL19894067 0.86 HCRTR2 (0.51) HCRTR2HCRTR1CYP3A4
Hydrochloric Acid SCHEMBL19893890 0.85 HCRTR2 (0.50) HCRTR2HCRTR1CYP3A4
SCHEMBL20212712 0.81 HCRTR2 (0.54) HCRTR2HCRTR1CYP3A4
SCHEMBL19894142 0.81 HCRTR2 (0.62) HCRTR2HCRTR1
Hydrochloric Acid SCHEMBL19894103 0.80 HCRTR2 (0.61) HCRTR2HCRTR1
SCHEMBL19903058 0.80 HCRTR2 (0.51) HCRTR2HCRTR1CYP3A4
SCHEMBL19903005 0.80 HCRTR2 (0.53) HCRTR2HCRTR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349270-A1 2,5-DISUBSTITUTED MORPHOLINE OREXIN RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-08-03 EP disclosed
WO-2010048013-A1 2,5-DISUBSTITUTED MORPHOLINE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-04-29 WO disclosed