SCHEMBL2358754

SCHEMBL2358754

Cc1ccc(-n2nccn2)c(C(=O)N2CCCCC2)c1

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 19/20 0.64
HCRTR1 O43613 17/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17539262 1.00 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL17501812 0.99 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL23018148 0.87 HCRTR2 (0.58) HCRTR2HCRTR1
SCHEMBL2356095 0.86 HCRTR2 (0.58) HCRTR2HCRTR1
SCHEMBL21443716 0.84 HCRTR2 (0.60) HCRTR2HCRTR1
SCHEMBL8209215 0.84 HCRTR2 (0.59) HCRTR2HCRTR1
SCHEMBL13106337 0.83 HCRTR1 (0.61) HCRTR2HCRTR1
SCHEMBL13733737 0.82 HCRTR2 (0.49) HCRTR2HCRTR1
SCHEMBL17502930 0.81 HCRTR2 (0.52) HCRTR2HCRTR1
SCHEMBL7911862 0.81 HCRTR2 (0.67) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350066-A1 2,5-DISUBSTITUTED PIPERIDINE OREXIN RECEPTOR ANTAGONISTS Merck Sharp & Dohme Corp. (US) 2011-08-03 EP claimed