SCHEMBL2356512

SCHEMBL2356512

COc1cc2nccc(Oc3ccc(NC(=O)c4cc(C5=CC=CCN5)cn(Cc5ccccc5)c4=O)nc3)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.69
PTK2B Q14289 7/20 0.61
PTK2 Q05397 2/20 0.61
MET P08581 9/20 0.55
AXL P30530 2/20 0.54
MERTK Q12866 1/20 0.54
EIF2AK3 Q9NZJ5 2/20 0.52
EIF2AK4 Q9P2K8 1/20 0.52
IGF1R P08069 1/20 0.52
KDR P35968 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL200000 0.86 SYK (0.75) SYKPTK2BPTK2METAXL
SCHEMBL200020 0.85 PTK2B (0.79) SYKPTK2BPTK2METAXL
SCHEMBL201489 0.85 SYK (0.68) SYKPTK2BPTK2METAXL
SCHEMBL199798 0.85 SYK (0.81) SYKPTK2BPTK2METAXL
SCHEMBL200792 0.85 SYK (0.73) SYKPTK2BPTK2METAXL
SCHEMBL199499 0.84 PTK2B (0.79) SYKPTK2BPTK2METAXL
SCHEMBL2356509 0.81 SYK (0.69) SYKPTK2BPTK2METAXL
SCHEMBL199512 0.79 SYK (0.63) SYKPTK2BPTK2METAXL
SCHEMBL199755 0.78 SYK (0.73) SYKPTK2BPTK2METAXL
SCHEMBL12993745 0.76 SYK (0.64) SYKPTK2BPTK2METAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349328-A1 METHODS FOR THE TREATMENT OF CANCER LUDWIG INSTITUTE FOR CANCER RESEARCH (US) 2011-08-03 EP claimed
WO-2010039248-A1 METHODS FOR THE TREATMENT OF CANCER LUDWIG INSTITUTE FOR CANCER RESEARCH (US) 2010-04-08 WO claimed