SCHEMBL23567650

SCHEMBL23567650

CCOC(=O)c1[nH]nc2c1C[C@@H]1C[C@]1(C)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.39
MAPK10 P53779 1/20 0.39
RIPK1 Q13546 1/20 0.39
HSD17B10 Q99714 2/20 0.37
PDE4D Q08499 1/20 0.36
MAPT P10636 2/20 0.34
KDM4E B2RXH2 4/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MEN1 O00255 1/20 0.34
ALOX15 P16050 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
ITK Q08881 3/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23567652 0.80 AURKA (0.38) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL23567665 0.77 ITK (0.47) AURKARIPK1MAPTKDM4EMEN1
SCHEMBL23565145 0.77 ITK (0.47) AURKARIPK1MAPTKDM4EMEN1
SCHEMBL25545776 0.77 ITK (0.47) AURKARIPK1MAPTKDM4EMEN1
SCHEMBL2471811 0.76 AURKA (0.43) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL19140049 0.75 AURKA (0.44) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL19140474 0.74 KDM4E (0.45) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL30587533 0.73 ALDH1A1 (0.45) AURKAMAPK10RIPK1HSD17B10MAPT
SCHEMBL30092714 0.73 AURKA (0.40) AURKAMAPK10RIPK1HSD17B10PDE4D
SCHEMBL4488956 0.72 AURKA (0.38) AURKAMAPK10RIPK1HSD17B10PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021124155-A1 BENZIMIDAZOLE DERIVATIVES PFIZER INC. (US) 2021-06-24 WO disclosed