SCHEMBL2358522

SCHEMBL2358522

CNC(C)C(=O)Nc1c(C)cc(-c2ccc(F)cc2)n(C(=O)N(CCc2ccccc2)CCc2ccccc2)c1=O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.36
KMT2A Q03164 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
XIAP P98170 6/20 0.35
BIRC2 Q13490 2/20 0.34
ELANE P08246 1/20 0.34
ASAH1 Q13510 5/20 0.34
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2358516 1.00 TACR1 (0.36) TACR1KMT2AHDAC6XIAPBIRC2
SCHEMBL4777094 0.78 CA12 (0.34) KMT2AHDAC6XIAPBIRC2ASAH1
SCHEMBL3852283 0.75 ELANE (0.42) XIAPELANE
SCHEMBL2358520 0.75 ELANE (0.42) XIAPELANE
SCHEMBL2209223 0.73 TP53 (0.39) HDAC6BIRC2ELANE
SCHEMBL2212581 0.73 ELANE (0.49) ELANE
SCHEMBL2212579 0.73 ELANE (0.49) ELANE
SCHEMBL2209218 0.73 TP53 (0.39) HDAC6BIRC2ELANE
SCHEMBL3832813 0.72 CA12 (0.38) KMT2AHDAC6BIRC2ELANE
SCHEMBL3830340 0.70 BIRC2 (0.37) XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989441-B2 Organic compounds NOVARTIS AG (CH) 2011-08-02 US claimed