SCHEMBL4777094

SCHEMBL4777094

CNC(C)C(=O)Nc1c(I)cc(-c2ccc(F)cc2)n(CC(=O)N(CCc2ccccc2)CCc2ccccc2)c1=O

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
HDAC6 Q9UBN7 1/20 0.33
BIRC2 Q13490 1/20 0.33
MMP2 P08253 1/20 0.33
XIAP P98170 4/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
ASAH1 Q13510 4/20 0.32
LMNA P02545 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2358520 0.85 ELANE (0.42) XIAP
SCHEMBL3852283 0.85 ELANE (0.42) XIAP
SCHEMBL2209223 0.83 TP53 (0.39) HDAC6BIRC2MMP2MAPTLMNA
SCHEMBL2209218 0.83 TP53 (0.39) HDAC6BIRC2MMP2MAPTLMNA
SCHEMBL4774566 0.79 CES2 (0.46) MAPTKMT2ALMNANPC1RAB9A
SCHEMBL2212581 0.79 ELANE (0.49)
SCHEMBL2212579 0.79 ELANE (0.49)
SCHEMBL3832813 0.79 CA12 (0.38) CA12CA1CA2CA4HDAC6
SCHEMBL2358516 0.78 TACR1 (0.36) HDAC6BIRC2XIAPKMT2AASAH1
SCHEMBL2358522 0.78 TACR1 (0.36) HDAC6BIRC2XIAPKMT2AASAH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902065-A2 CYCLIC AMIDE DERIVATIVES INHIBITORS OF THE INHIBITOR OF APOPTOSIS PROTEINS, THEIR PREPARATION, AND THEIR USE Novartis AG (CH) 2008-03-26 EP claimed
WO-2006133147-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2006-12-14 WO claimed