SCHEMBL2360175

SCHEMBL2360175

CCC1CN(CCOc2cc(C)n(-c3ccc(Cl)c(Cl)c3)n2)CCN1C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 20/20 0.66
KCNH2 Q12809 3/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17530637 0.83 SIGMAR1 (0.82) SIGMAR1KCNH2
Oxalic Acid SCHEMBL4511455 0.81 SIGMAR1 (0.69) SIGMAR1KCNH2
SCHEMBL467173 0.80 SIGMAR1 (0.83) SIGMAR1KCNH2
SCHEMBL19988158 0.80 SIGMAR1 (0.85) SIGMAR1KCNH2
Oxalic Acid SCHEMBL4521956 0.80 SIGMAR1 (0.79) SIGMAR1KCNH2
SCHEMBL466869 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL29558224 0.80 SIGMAR1 (1.00) SIGMAR1KCNH2
Hydrochloric Acid SCHEMBL1897332 0.79 SIGMAR1 (0.98) SIGMAR1KCNH2
SCHEMBL467027 0.79 SIGMAR1 (1.00) SIGMAR1KCNH2
SCHEMBL4560092 0.79 SIGMAR1 (0.78) SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2571501-B1 SIGMA LIGANDS FOR THE PREVENTION AND/OR TREATMENT OF EMESIS INDUCED BY CHEMOTHERAPY OR RADIOTHERAPY ESTEVE LABOR DR (ES) 2016-03-02 EP claimed
EP-1781618-B1 SIGMA RECEPTOR INHIBITORS ESTEVE LABOR DR (ES) 2012-10-03 EP claimed
WO-2011095585-A1 SIGMA LIGANDS FOR POTENTIATING THE ANALGESIC EFFECT OF OPIOIDS AND OPIATES IN POST-OPERATIVE PAIN AND ATTENUATING THE DEPENDENCY THEREOF LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2011-08-11 WO claimed
WO-2011095585-A1 SIGMA LIGANDS FOR POTENTIATING THE ANALGESIC EFFECT OF OPIOIDS AND OPIATES IN POST-OPERATIVE PAIN AND ATTENUATING THE DEPENDENCY THEREOF LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2011-08-11 WO disclosed