SCHEMBL2361404

SCHEMBL2361404

CC1Cc2c([nH]c3ccc(F)cc23)C2(CCC(C(c3ccc(Cl)cc3)[As](C)C)CC2)O1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.54
OGFRL1 Q5TC84 7/20 0.54
CYP2C9 P11712 2/20 0.41
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
CFTR P13569 1/20 0.35
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
VPS4B O75351 1/20 0.33
VCP P55072 1/20 0.33
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
HTR2A P28223 2/20 0.31
HTR2B P41595 2/20 0.31
HTR2C P28335 1/20 0.31
DRD2 P14416 2/20 0.31
SLC6A4 P31645 2/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL699747 0.86 OPRM1 (0.58) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL698663 0.81 OPRM1 (0.61) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL700139 0.78 OPRM1 (0.67) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL700959 0.77 OPRM1 (0.61) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL699857 0.76 OPRM1 (0.58) OPRM1OGFRL1CYP2C9HTR2AHTR2B
SCHEMBL699255 0.76 OPRM1 (0.64) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL699418 0.75 OPRM1 (0.57) OPRM1OGFRL1OPRD1OPRK1OPRL1
SCHEMBL706789 0.74 OPRM1 (0.56) OPRM1OGFRL1CYP2C9OPRD1OPRK1
SCHEMBL699256 0.72 OPRM1 (0.62) OPRM1OGFRL1OPRD1OPRK1OPRL1
SCHEMBL699742 0.71 OPRM1 (0.55) OPRM1OGFRL1CYP2C9OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010531-B1 SPIROCYCLIC CYCLOHEXANE DERIVATIVES WITH ANALGESIC PROPERTIES GRUENENTHAL GMBH (DE) 2011-08-17 EP disclosed