SCHEMBL23616222

SCHEMBL23616222

CC(C)CC(NC(=O)[C@H](CCc1ccccc1)NC(=O)CN1CCOCC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)C1(C)CC1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 17/20 0.84
PSMB9 P28065 3/20 0.84
PSMB8 P28062 3/20 0.84
PSMB10 P40306 3/20 0.84
PSMB2 P49721 3/20 0.84
CYP3A4 P08684 2/20 0.84
CYP3A5 P20815 2/20 0.84
CYP3A7 P24462 2/20 0.84
CYP3A43 Q9HB55 2/20 0.84
PSMB11 A5LHX3 1/20 0.84
PSMD11 O00231 1/20 0.84
PSMD12 O00232 1/20 0.84
PSMD14 O00487 1/20 0.84
PSMA7 O14818 1/20 0.84
PSMD3 O43242 1/20 0.84
CTSB P07858 1/20 0.84
PSMC3 P17980 1/20 0.84
PSMB1 P20618 1/20 0.84
PSMA1 P25786 1/20 0.84
PSMA2 P25787 1/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL84978 1.00 PSMB5 (0.84) PSMB5PSMB9PSMB8PSMB10PSMB2
SCHEMBL9909637 0.93 PSMB5 (0.74) PSMB5PSMB9PSMB8PSMB10PSMB2
SCHEMBL8267515 0.93 PSMB5 (0.72) PSMB5PSMB9PSMB8PSMB10PSMB2
SCHEMBL84929 0.92 PSMB5 (0.73) PSMB5PSMB9PSMB8PSMB10PSMB2
SCHEMBL84985 0.91 PSMB5 (0.70) PSMB5PSMB9PSMB8PSMB10PSMB2
Carfilzomib SCHEMBL23616374 0.91 PSMB5 (1.00) PSMB5PSMB9PSMB8PSMB10PSMB2
Carfilzomib SCHEMBL20533771 0.91 PSMB5 (1.00) PSMB5PSMB9PSMB8PSMB10PSMB2
Carfilzomib SCHEMBL25438395 0.91 PSMB5 (1.00) PSMB5PSMB9PSMB8PSMB10PSMB2
Carfilzomib SCHEMBL21035706 0.91 PSMB5 (1.00) PSMB5PSMB9PSMB8PSMB10PSMB2
Carfilzomib SCHEMBL21036025 0.91 PSMB5 (1.00) PSMB5PSMB9PSMB8PSMB10PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3297678-B1 AN IMPROVED PROCESSES FOR THE PREPARATION OF CARFILZOMIB OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF LAURUS LABS LTD (IN) 2021-07-07 EP disclosed