SCHEMBL2362084

SCHEMBL2362084

COCc1cc(C(N)=O)c(-c2ccc[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.37
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 2/20 0.32
GAA P10253 2/20 0.32
TYK2 P29597 1/20 0.32
NAPRT Q6XQN6 1/20 0.31
MAPT P10636 2/20 0.31
TSHR P16473 1/20 0.31
ACVR1 Q04771 1/20 0.31
SCN9A Q15858 1/20 0.31
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
THRB P10828 1/20 0.30
BLM P54132 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
IKBKB O14920 1/20 0.30
PRSS1 P07477 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2349673 0.83 CYP1A1 (0.37) CYP3A4NPC1RAB9ATYK2L3MBTL1
SCHEMBL2128919 0.74 CYP3A4 (0.52) CYP3A4TYK2NAPRTL3MBTL1IKBKB
SCHEMBL2364691 0.73 ICMT (0.44) CYP3A4L3MBTL1CD274
SCHEMBL2354432 0.72 KDM4E (0.40) CYP3A4NPC1RAB9AKDM4EALDH1A1
SCHEMBL2350724 0.72 NAPRT (0.43) CYP3A4KDM4EALDH1A1NAPRTL3MBTL1
SCHEMBL2363082 0.70 HTR2A (0.44) CYP3A4KDM4EALDH1A1GAAL3MBTL1
SCHEMBL2363467 0.70 CYP3A4 (0.43) CYP3A4KDM4EALDH1A1GAAMAPT
SCHEMBL2354510 0.70 CYP3A4 (0.41) CYP3A4KDM4EGAAL3MBTL1
SCHEMBL3316087 0.70 MAP4K1 (0.38) CYP3A4NAPRTMAPTMEN1KMT2A
SCHEMBL2362083 0.70 PLK1 (0.38) CYP3A4KDM4EALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350007-A1 HETEROCYCLIC ANTIVIRAL ARYLPYRIDONE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-08-03 EP disclosed
WO-2010049331-A1 HETEROCYCLIC ANTIVIRAL ARYLPYRIDONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-05-06 WO disclosed