SCHEMBL23623116

SCHEMBL23623116

COC(=O)c1cnc(C)c(Cl)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.43
MRGPRX4 Q96LA9 2/20 0.41
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
LCK P06239 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3710244 0.86 MAPK1 (0.43) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL30420441 0.86 MAPK1 (0.43) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL17008727 0.85 MAPK1 (0.46) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL30019960 0.85 MAPK1 (0.46) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL12066239 0.83 MAPK1 (0.47) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL7454206 0.81 MAPK1 (0.46) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL1105939 0.81 ALDH1A1 (0.46) MAPK1SMN1; SMN2L3MBTL1ALDH1A1KDM4E
SCHEMBL30773331 0.81 MAPK1 (0.42) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL24369506 0.81 MAPK1 (0.42) MAPK1MRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL23623115 0.79 SMN1; SMN2 (0.38) MAPK1NPC1RAB9ASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116601158-A Modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-08-15 CN disclosed
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed
WO-2021138434-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY IFM DUE, INC. (US) 2021-07-08 WO disclosed