SCHEMBL2362779

SCHEMBL2362779

CON1CCC2(CC1)NC(=O)C(c1cc(-c3ccc(F)cc3)ccc1C)=C2O

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACACB O00763 13/20 0.59
ACACA Q13085 13/20 0.59
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
OTUD7B Q6GQQ9 2/20 0.32
STK10 O94804 1/20 0.32
SLK Q9H2G2 1/20 0.32
SSTR5 P35346 1/20 0.32
KCNH2 Q12809 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2362487 0.91 ACACB (0.64) ACACBACACA
SCHEMBL11888077 0.90 ACACB (0.73) ACACBACACA
SCHEMBL2361925 0.89 ACACB (0.56) ACACBACACAOTUD7BSTK10SLK
SCHEMBL29735375 0.86 ACACB (0.53) ACACBACACA
SCHEMBL249181 0.86 ACACB (0.53) ACACBACACA
SCHEMBL12540243 0.86 ACACB (0.79) ACACBACACACNR1CNR2TNKS2
SCHEMBL12256245 0.85 ACACB (0.45) ACACBACACACNR1CNR2
SCHEMBL12029732 0.85 ACACB (0.60) ACACBACACATNKS2
SCHEMBL12456400 0.85 ACACB (0.54) ACACBACACAKCNH2TNKS2
SCHEMBL2362922 0.84 ACACB (0.44) ACACBACACASSTR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9809542-B2 Spiroheterocyclically substituted tetramic acid derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-11-07 US disclosed
US-9809542-B2 Spiroheterocyclically substituted tetramic acid derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-11-07 US disclosed
US-9809542-B2 Spiroheterocyclically substituted tetramic acid derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2017-11-07 US disclosed
EP-2534147-B1 SPIROHETEROCYCLIC-SUBSTITUTED TETRAMIC ACID DERIVATIVES BAYER IP GMBH (DE) 2015-06-17 EP disclosed
EP-2534147-A1 SPIROHETEROCYCLICAL SUBSTITUTED TETRAMIC ACID DERIVATIVES Bayer Intellectual Property GmbH (DE) 2012-12-19 EP disclosed
US-20110230351-A1 Spiroheterocyclically Substituted Tetramic Acid Derivatives BAYER CROPSCIENCE AG (DE) 2011-09-22 US disclosed
US-20110230351-A1 Spiroheterocyclically Substituted Tetramic Acid Derivatives BAYER CROPSCIENCE AG (DE) 2011-09-22 US disclosed
US-20110230351-A1 Spiroheterocyclically Substituted Tetramic Acid Derivatives BAYER CROPSCIENCE AG (DE) 2011-09-22 US disclosed
WO-2011098443-A1 SPIROHETEROCYCLICAL SUBSTITUTED TETRAMIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2011-08-18 WO disclosed
WO-2011098443-A1 SPIROHETEROCYCLICAL SUBSTITUTED TETRAMIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2011-08-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110230351-A1 Spiroheterocyclically Substituted Tetramic Acid Derivatives AGXT, PTPRG, WIZ ACACB 904/4885ACACA 192/4885CNR1 3516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.