SCHEMBL23628480

SCHEMBL23628480

NS(=O)(=O)c1ccc(C(=O)N2CC3=C(CNC3)C2)c(F)c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 16/20 0.57
CA1 P00915 10/20 0.46
CA9 Q16790 6/20 0.46
CA12 O43570 4/20 0.46
CA7 P43166 4/20 0.46
CA14 Q9ULX7 4/20 0.46
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
GAA P10253 2/20 0.41
SLC6A9 P48067 1/20 0.38
CPS1 P31327 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL18668453 0.99 CA2 (0.56) CA2CA1CA9CA12CA7
Hydrochloric Acid SCHEMBL22205231 0.99 CA2 (0.56) CA2CA1CA9CA12CA7
SCHEMBL23628462 0.86 CA2 (0.58) CA2CA1CA9CA12CA7
Hydrochloric Acid SCHEMBL22205236 0.83 CA2 (0.47) CA2CA1CA9CA12CA7
SCHEMBL23628502 0.80 CA2 (0.66) CA2CA1CA12CA7
SCHEMBL28723643 0.80 CA2 (0.52) CA2CA1CA9CA12CA7
SCHEMBL29571991 0.80 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL23628490 0.79 CA2 (0.49) CA2CA1CA9CA12CA7
SCHEMBL18668482 0.79 CA2 (0.56) CA2CA1CA9CA12CA7
SCHEMBL20502378 0.77 CA2 (0.59) CA2CA1CA9CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353178-B1 BICYCLIC COMPOUNDS AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2021-07-14 EP disclosed