SCHEMBL23629627

SCHEMBL23629627

CCOC(=O)C1(OCC)C=Cc2ccccc2N1I

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 2/20 0.38
P2RX4 Q99571 5/20 0.36
P2RX1 P51575 2/20 0.36
P2RX3 P56373 2/20 0.36
BCHE P06276 1/20 0.36
PTBP1 P26599 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
P2RX7 Q99572 1/20 0.36
OPRM1 P35372 5/20 0.35
OPRD1 P41143 3/20 0.35
OPRK1 P41145 3/20 0.35
SLC22A1 O15245 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18601369 0.85 P2RX4 (0.36) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL31350302 0.74 P2RX4 (0.41) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL2204621 0.73 SMN1; SMN2 (0.45) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL30643764 0.73 P2RX4 (0.38) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL11168819 0.73 P2RX4 (0.38) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL10743523 0.72 SMN1; SMN2 (0.47) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL30250427 0.68 BRD4 (0.40) SMN1; SMN2MAPK1OPRM1OPRD1OPRK1
SCHEMBL6991005 0.68 BRD4 (0.40) SMN1; SMN2MAPK1OPRM1OPRD1OPRK1
Propionic Acid SCHEMBL31424601 0.68 SMN1; SMN2 (0.43) SMN1; SMN2LMNAMAPK1P2RX4P2RX1
SCHEMBL11412073 0.67 P2RX4 (0.71) SMN1; SMN2LMNAMAPK1P2RX4P2RX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3847166-A1 POLYCYCLIC AMIDES AS CYTOTOXIC AGENTS Femtogenix Limited (GB) 2021-07-14 EP disclosed