SCHEMBL23632012

SCHEMBL23632012

O=C(O)c1ccc(Cn2ncc3cc(F)ccc32)cc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.50
AGTR2 P50052 2/20 0.50
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
EPHX2 P34913 1/20 0.47
PPARG P37231 1/20 0.47
CPT1A P50416 1/20 0.46
CPT1B Q92523 1/20 0.46
RECQL P46063 1/20 0.46
ENPP2 Q13822 1/20 0.45
PTGER4 P35408 3/20 0.45
HDAC2 Q92769 2/20 0.45
CCR2 P41597 1/20 0.44
KMO O15229 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HDAC1 Q13547 1/20 0.43
TP53 P04637 1/20 0.43
HCAR3 P49019 1/20 0.43
SMO Q99835 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30614175 0.92 EPHX2 (0.47) AGTR1AGTR2EPHX2PPARGRECQL
SCHEMBL698761 0.92 EPHX2 (0.47) AGTR1AGTR2EPHX2PPARGRECQL
SCHEMBL30614172 0.87 EPHX2 (0.49) AGTR1AGTR2HTR2AHTR2CEPHX2
SCHEMBL25414085 0.87 EPHX2 (0.49) AGTR1AGTR2HTR2AHTR2CEPHX2
SCHEMBL23632579 0.85 CYP11B1 (0.56) HTR2AHTR2CEPHX2PPARGHDAC2
SCHEMBL16595434 0.85 EPHX2 (0.46) HTR2AHTR2CEPHX2PPARGRECQL
SCHEMBL27787592 0.84 RECQL (0.46) EPHX2PPARGRECQLPTGER4KMO
SCHEMBL6840434 0.84 BRD4 (0.49) RECQLENPP2PTGER4KMOTP53
SCHEMBL31633189 0.84 EPHX2 (0.62) EPHX2PPARGRECQLPTGER4HCAR3
SCHEMBL6840422 0.83 P2RY14 (0.47) HTR2AHTR2CEPHX2PPARGHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072542-B ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
WO-2021139595-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed
CN-113072542-A ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed