SCHEMBL23632579

SCHEMBL23632579

COC(=O)c1ccc(Cn2ncc3cc(F)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56
GAA P10253 1/20 0.51
RAB9A P51151 1/20 0.51
FAAH O00519 1/20 0.48
EPHX2 P34913 2/20 0.48
PPARG P37231 2/20 0.48
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
TP53 P04637 2/20 0.47
POLB P06746 1/20 0.47
HDAC2 Q92769 1/20 0.46
P2RX3 P56373 1/20 0.44
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25408602 0.88 EPHX2 (0.50) CYP11B1CYP11B2GAARAB9AFAAH
SCHEMBL25413272 0.86 BRD4 (0.51) CYP11B1CYP11B2GAARAB9AFAAH
SCHEMBL30614188 0.86 BRD4 (0.51) CYP11B1CYP11B2GAARAB9AFAAH
SCHEMBL31632909 0.85 EPHX2 (0.61) CYP11B1CYP11B2EPHX2PPARGEGFR
SCHEMBL23632012 0.85 AGTR1 (0.50) EPHX2PPARGHTR2AHTR2CTP53
SCHEMBL16596018 0.84 EPHX2 (0.47) CYP11B1CYP11B2EPHX2PPARGHDAC2
SCHEMBL1418153 0.83 HDAC6 (0.51) GAARAB9AFAAHEPHX2PPARG
SCHEMBL25411989 0.83 GAA (0.48) CYP11B1CYP11B2GAARAB9AFAAH
SCHEMBL16056414 0.83 CYP11B1 (0.50) CYP11B1CYP11B2GAARAB9AEPHX2
SCHEMBL3724300 0.83 RECQL (0.60) GAARAB9AFAAHMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072542-B ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业股份有限公司 2024-04-05 CN disclosed
WO-2021139595-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed
CN-113072542-A ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed