SCHEMBL23633131

SCHEMBL23633131

CCC(F)(F)OC[C@@H]1C[C@H](Oc2ccc(C(F)(F)F)cc2)CN1c1ccc(C(=O)O)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 1/20 0.41
ACACB O00763 1/20 0.40
EPHX2 P34913 1/20 0.37
GRM4 Q14833 1/20 0.36
TACR1 P25103 1/20 0.35
TACR3 P29371 1/20 0.35
LIPG Q9Y5X9 2/20 0.35
LPL P06858 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
GCGR P47871 2/20 0.35
GCG P01275 1/20 0.35
RET P07949 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.34
ADRB2 P07550 1/20 0.34
SCN9A Q15858 2/20 0.34
PPARD Q03181 1/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23632833 1.00 PRKAA2 (0.41) PRKAA2ACACBEPHX2GRM4TACR1
SCHEMBL28592571 0.92 ACACB (0.41) PRKAA2ACACBGRM4TACR1TACR3
SCHEMBL30065111 0.92 ACACB (0.41) PRKAA2ACACBGRM4TACR1TACR3
SCHEMBL23632467 0.91 PRKAA2 (0.42) PRKAA2ACACBEPHX2GRM4TACR1
SCHEMBL23632822 0.90 ACACB (0.37) PRKAA2ACACBEPHX2GRM4LIPG
SCHEMBL23632578 0.90 ACACB (0.37) PRKAA2ACACBEPHX2GRM4LIPG
SCHEMBL23632613 0.87 EPHX2 (0.42) EPHX2LIPGADRB2LTA4H
SCHEMBL23632256 0.87 EPHX2 (0.42) EPHX2LIPGADRB2LTA4H
SCHEMBL23632629 0.86 PRKAA2 (0.41) PRKAA2ACACBEPHX2GRM4TACR1
SCHEMBL23632193 0.86 PRKAA2 (0.41) PRKAA2ACACBEPHX2GRM4TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021139599-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed