SCHEMBL23632578

SCHEMBL23632578

CCC(F)(F)OC[C@@H]1C[C@@H](Oc2ccc(C(F)(F)F)cc2)CN1c1ncc(C(=O)O)cn1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.37
SCN9A Q15858 4/20 0.36
EPHX2 P34913 2/20 0.36
LIPG Q9Y5X9 4/20 0.36
LPL P06858 1/20 0.36
RBP4 P02753 1/20 0.35
PRKAA2 P54646 1/20 0.35
GRM4 Q14833 1/20 0.35
LIPC P11150 1/20 0.34
LIPE Q05469 1/20 0.34
FFAR1 O14842 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23632822 1.00 ACACB (0.37) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL23632206 0.91 EPHX2 (0.39) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL23632894 0.91 EPHX2 (0.39) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL28601527 0.91 ACACB (0.44) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL23632833 0.90 PRKAA2 (0.41) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL23633131 0.90 PRKAA2 (0.41) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL23632613 0.86 EPHX2 (0.42) EPHX2LIPGLIPCLIPEFFAR1
SCHEMBL23632256 0.86 EPHX2 (0.42) EPHX2LIPGLIPCLIPEFFAR1
SCHEMBL23632735 0.85 ACACB (0.38) ACACBSCN9AEPHX2LIPGLPL
SCHEMBL28529263 0.85 RBP4 (0.38) ACACBRBP4GRM4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021139599-A1 RORγT INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 东莞市东阳光新药研发有限公司 2021-07-15 WO disclosed
CN-113072476-A ROR gamma t inhibitor and preparation method and application thereof 广东东阳光药业有限公司 2021-07-06 CN disclosed