SCHEMBL2364480

SCHEMBL2364480

COc1cccc(-c2ccc(C(Oc3cc(-c4ccc(CC(N)C(=O)O)cc4)nc(N)n3)C(F)(F)F)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 20/20 1.00
TPH2 Q8IWU9 11/20 1.00
ADORA3 P0DMS8 2/20 0.55
SLC6A2 P23975 2/20 0.55
AGTR1 P30556 2/20 0.55
SLC6A4 P31645 2/20 0.55
CCKAR P32238 2/20 0.55
SLC6A3 Q01959 2/20 0.55
F2 P00734 1/20 0.55
ESR1 P03372 1/20 0.55
DRD1 P21728 1/20 0.55
PTGS1 P23219 1/20 0.55
PTGS2 P35354 1/20 0.55
DRD3 P35462 1/20 0.55
MLNR O43193 1/20 0.47
NR3C1 P04150 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
MC3R P41968 1/20 0.47
HTR3A P46098 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL308718 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL29391423 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL308719 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL13878219 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL870345 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL870344 1.00 TPH1 (1.00) TPH1TPH2ADORA3SLC6A2AGTR1
Fumaric Acid SCHEMBL2927924 0.96 TPH1 (0.93) TPH1TPH2ADORA3SLC6A2AGTR1
Maleic Acid SCHEMBL2720175 0.96 TPH1 (0.93) TPH1TPH2ADORA3SLC6A2AGTR1
Fumaric Acid SCHEMBL2927928 0.96 TPH1 (0.93) TPH1TPH2ADORA3SLC6A2AGTR1
SCHEMBL12128916 0.94 TPH1 (0.89) TPH1TPH2ADORA3SLC6A2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113462728-B Method for preparing (R) -1- (4-bromophenyl) -2, 2-trifluoroethanol by using starwheel head yeast 浙江工业大学 2024-06-07 CN disclosed
CN-113462728-A Method for preparing (R) -1- (4-bromophenyl) -2,2, 2-trifluoroethanol by using Verticillium terrestris 浙江工业大学 2021-10-01 CN disclosed
EP-2358685-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED PHENYLALANINES Lexicon Pharmaceuticals, Inc. (US) 2011-08-24 EP disclosed
CN-101932563-A Solid forms of (s)-2-amino-3-(4-(2-amino-6-((r)-2,2,2-trifluoro-1-(3'-methoxybiphenyl-4-yl)ethoxy)pyrimidin-4-yl)phenyl)propanoic acid and methods of their use LEXICON PHARMACEUTICALS INC 2010-12-29 CN disclosed
WO-2010047712-A1 PROCESS FOR THE PREPARATION OF SUBSTITUTED PHENYLALANINES LEXICON PHARMACEUTICALS, INC. (US) 2010-04-29 WO disclosed