SCHEMBL23648147

SCHEMBL23648147

O=C1Nc2c(Br)cc(F)cc2C12CC2

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
PGR P06401 5/20 0.34
AKR1A1 P14550 2/20 0.31
AKR1B1 P15121 2/20 0.31
KMT2A Q03164 1/20 0.31
AKR1B10 O60218 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30858557 0.79 KMT2A (0.41) ALDH1A1HTTMAPTCYP1A2CYP2C19
SCHEMBL31492406 0.79 DAO (0.35) ALDH1A1LMNATP53HTTPGR
SCHEMBL4813479 0.76 PGR (0.41) ALDH1A1LMNATP53HTTPGR
SCHEMBL4779068 0.74 PGR (0.32) ALDH1A1LMNATP53HTTPGR
SCHEMBL16849905 0.73 PDE7A (0.35) ALDH1A1LMNATP53HTTMAPT
SCHEMBL31492415 0.73 PGR (0.33) ALDH1A1LMNATP53HTTPGR
SCHEMBL3522002 0.73 PGR (0.67) PGR
SCHEMBL30224301 0.72 PGR (0.32) PGR
SCHEMBL23994828 0.72 PGR (0.32) PGR
SCHEMBL23647999 0.70 PGR (0.34) PGRAKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4090660-A1 QUINOXALINE DERIVATIVES Grünenthal GmbH (DE) 2022-11-23 EP disclosed
WO-2021144439-A1 QUINOXALINE DERIVATIVES Grünenthal GmbH (DE) 2021-07-22 WO disclosed
WO-2021144439-A1 QUINOXALINE DERIVATIVES Grünenthal GmbH (DE) 2021-07-22 WO disclosed