SCHEMBL23648792

SCHEMBL23648792

CSc1ncc2c(n1)N(C)C(=O)N(c1cc(Br)ccc1C)C2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 2/20 0.60
TNK2 Q07912 10/20 0.43
MAP4K2 Q12851 10/20 0.43
BMX P51813 9/20 0.43
ABL1 P00519 4/20 0.43
LCK P06239 1/20 0.43
FES P07332 1/20 0.43
RET P07949 1/20 0.43
PDGFRB P09619 1/20 0.43
KIT P10721 1/20 0.43
FGFR1 P11362 1/20 0.43
SRC P12931 1/20 0.43
PDGFRA P16234 1/20 0.43
FLT1 P17948 1/20 0.43
FGFR3 P22607 1/20 0.43
EPHA3 P29320 1/20 0.43
KDR P35968 1/20 0.43
EPHB4 P54760 1/20 0.43
TEK Q02763 1/20 0.43
KARS1 Q15046 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6620382 0.84 FGFR4 (0.61) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL1521938 0.80 FGFR4 (0.56) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL6621872 0.79 FGFR4 (0.62) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL1521396 0.76 FGFR4 (0.52) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL6620598 0.76 FGFR4 (0.71) FGFR4TNK2MAP4K2ABL1FGFR1
SCHEMBL15412943 0.75 FGFR4 (1.00) FGFR4BMXFGFR1FGFR3KDR
SCHEMBL5229018 0.73 FGFR4 (0.61) FGFR4LCKFGFR1FGFR3KDR
SCHEMBL6618207 0.73 FGFR4 (0.61) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL1521583 0.73 FGFR4 (0.55) FGFR4TNK2MAP4K2BMXABL1
SCHEMBL3573608 0.73 FGFR4 (0.55) FGFR4TNK2MAP4K2BMXABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021145520-A1 7-AMINO-3,4-DIHYDROPYRIMIDOPYRIMIDIN-2-ONE DERIVATIVE HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES AND THERAPEUTIC PHARMACEUTICAL COMPOSITION COMPRISING SAME 한국과학기술연구원 2021-07-22 WO disclosed
WO-2021145520-A1 7-AMINO-3,4-DIHYDROPYRIMIDOPYRIMIDIN-2-ONE DERIVATIVE HAVING INHIBITORY ACTIVITY FOR PROTEIN KINASES AND THERAPEUTIC PHARMACEUTICAL COMPOSITION COMPRISING SAME 한국과학기술연구원 2021-07-22 WO disclosed