SCHEMBL2364951

SCHEMBL2364951

CS(=O)(=O)c1ccc(NC(=O)c2ccccc2C(F)(F)F)cc1NC(=O)c1csc2c(N)ncnc12

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BRAF P15056 8/20 0.44
PTGS1 P23219 1/20 0.43
ERN1 O75460 1/20 0.43
CSF1R P07333 9/20 0.42
PTPRC P08575 1/20 0.41
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
RAF1 P04049 6/20 0.41
CYP2C9 P11712 1/20 0.41
DDR2 Q16832 5/20 0.40
DDR1 Q08345 4/20 0.40
PTGES O14684 1/20 0.40
FGFR1 P11362 1/20 0.40
KDR P35968 1/20 0.40
TEK Q02763 1/20 0.40
MELK Q14680 1/20 0.40
GRM4 Q14833 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2312969 0.88 RAF1 (0.48) BRAFPTGS1CSF1RAURKARAF1
SCHEMBL2364955 0.86 CSF1R (0.47) BRAFERN1CSF1RRAF1CYP2C9
SCHEMBL2364506 0.82 CSF1R (0.47) BRAFERN1CSF1RRAF1CYP2C9
SCHEMBL2233855 0.77 GRM4 (0.54) BRAFERN1CSF1RRAF1CYP2C9
SCHEMBL2359166 0.77 BRAF (0.46) BRAFERN1CSF1RRAF1CYP2C9
SCHEMBL12433866 0.75 CSF1R (0.53) BRAFCSF1RRAF1DDR2DDR1
SCHEMBL2314140 0.75 CSF1R (0.52) BRAFCSF1RAURKARAF1DDR2
SCHEMBL2356829 0.74 RAF1 (0.52) BRAFERN1CSF1RRAF1DDR2
SCHEMBL2313222 0.74 CSF1R (0.66) BRAFCSF1RRAF1CYP2C9DDR2
SCHEMBL2310995 0.74 BRAF (0.54) BRAFCSF1RAURKARAF1DDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2528925-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES Hanmi Science Co., Ltd. (KR) 2012-12-05 EP disclosed
WO-2011093684-A2 THIENO[3,2-d]PYRIMIDINE DERIVATIVES HAVING INHIBITORY ACTIVITY ON PROTEIN KINASES HANMI HOLDINGS CO., LTD. (KR) 2011-08-04 WO disclosed