SCHEMBL23653149

SCHEMBL23653149

COc1cc(C#N)cc(N)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
CYP3A4 P08684 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 1/20 0.38
AR P10275 3/20 0.38
HPGDS O60760 1/20 0.37
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
S100B P04271 1/20 0.36
ALOX12 P18054 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14871817 0.81 AR (0.40) ALDH1A1KDM4EUSP2ARHPGDS
SCHEMBL16122060 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EUSP2ARHPGDS
SCHEMBL1116020 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EUSP2CYP3A4L3MBTL1
SCHEMBL16072320 0.79 AR (0.45) ALDH1A1KDM4EUSP2ARHPGDS
SCHEMBL1496436 0.79 AR (0.42) ALDH1A1KDM4EUSP2CYP3A4L3MBTL1
SCHEMBL17522205 0.79 POLB (0.38) ALDH1A1KDM4EUSP2POLBAR
SCHEMBL7927109 0.78 ALDH1A1 (0.47) ALDH1A1KDM4EUSP2CYP3A4L3MBTL1
SCHEMBL17744575 0.78 TTR (0.44) ALDH1A1KDM4EUSP2CYP3A4L3MBTL1
SCHEMBL29104000 0.78 ALDH1A1 (0.41) ALDH1A1KDM4EUSP2CYP3A4L3MBTL1
SCHEMBL18112970 0.78 MEN1 (0.44) ALDH1A1KDM4EUSP2L3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3943087-A1 HETEROARYL COMPOUNDS AND USES THEREOF Celgene CAR LLC (BM) 2022-01-26 EP disclosed
EP-2968337-B1 HETEROARYL COMPOUNDS AND USES THEREOF CELGENE CAR LLC (BM) 2021-07-21 EP disclosed