SCHEMBL23653236

SCHEMBL23653236

CNc1ccccc1Nc1ncc2c(n1)N(C)C(=O)N(c1c(Cl)cccc1Cl)C2

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 14/20 0.74
LCK P06239 1/20 0.59
MAPK14 Q16539 1/20 0.59
FGFR1 P11362 2/20 0.49
SIK2 Q9H0K1 2/20 0.45
CSF1R P07333 1/20 0.45
SIK1 P57059 1/20 0.45
SIK3 Q9Y2K2 1/20 0.45
TNK2 Q07912 2/20 0.42
MAP4K2 Q12851 2/20 0.42
ABL1 P00519 1/20 0.41
FGFR2 P21802 1/20 0.41
FGFR3 P22607 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16072330 0.90 FGFR4 (0.71) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL21860438 0.89 FGFR4 (0.81) FGFR4LCKMAPK14FGFR1TNK2
SCHEMBL6622549 0.87 LCK (0.69) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL16071751 0.85 FGFR4 (1.00) FGFR4LCKMAPK14FGFR1FGFR2
SCHEMBL6620907 0.82 LCK (0.68) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL23653237 0.81 FGFR4 (0.91) FGFR4FGFR1FGFR2FGFR3
SCHEMBL6618406 0.81 FGFR4 (0.60) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL6619138 0.80 LCK (0.74) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL6620252 0.80 MAPK14 (0.66) FGFR4LCKMAPK14FGFR1SIK2
SCHEMBL6619141 0.78 FGFR4 (0.57) FGFR4LCKMAPK14FGFR1TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968337-B1 HETEROARYL COMPOUNDS AND USES THEREOF CELGENE CAR LLC (BM) 2021-07-21 EP disclosed