SCHEMBL23655441

SCHEMBL23655441

Cc1cnc(N)c(C#CSI)c1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.46
NOS2 P35228 3/20 0.46
NOS1 P29475 2/20 0.46
CYP2A6 P11509 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20382081 0.79
SCHEMBL18053335 0.78 NOS3 (0.52) NOS3NOS2NOS1CYP2A6
SCHEMBL1713842 0.77 NOS3 (0.50) NOS3NOS2NOS1CYP2A6
SCHEMBL20245056 0.74 CSF1R (0.43)
SCHEMBL13204736 0.74 NOS3 (0.47) NOS3NOS2NOS1CYP2A6
SCHEMBL4877753 0.72 NOS3 (0.54) NOS3NOS2NOS1CYP2A6
SCHEMBL31695297 0.72 NOS3 (0.54) NOS3NOS2NOS1CYP2A6
SCHEMBL625135 0.72 NOS3 (0.54) NOS3NOS2NOS1CYP2A6
SCHEMBL6488811 0.71 MAPT (0.46) NOS3NOS2NOS1
SCHEMBL24630011 0.69 GAA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3851437-A2 METHODS OF PREPARING 1H-PYRROLO[2,3-B]PYRIDINE DERIVATES Vertex Pharmaceuticals Incorporated (US) 2021-07-21 EP disclosed
WO-2017133667-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA THEREOF SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed